3
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T11486 | GSK2807 Trifluoroacetate | Histone Methyltransferase | |
GSK2807 Trifluoroacetate is a selective and SAM-competitive inhibitor of SMYD3 (Ki: 14 nM; IC50: 130 nM). | |||
T69738 | GSK-2807 free base | ||
GSK2807 is a potent and selective, SAM-competitive inhibitor of SMYD3 (Ki = 14 nM). GSK2807 bridges the gap between the SAM-binding pocket and the substrate lysine tunnel of SMYD3. GSK2807 may be useful for cancer trea... | |||
T69737 | SCH-79687 | ||
SCH-79687 is a histamine antagonist selective for the H3 subtype. This H3 antagonist may play a role in allergic rhinitis. |